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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T81662 | N-Nitrosodicyclohexylamine | NDCHA | Androgen Receptor |
N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in opposition to 5α-dihydrotestosterone and reducing AR protein levels [1... | |||
T35668 | Neoaureothin | ||
Neoaureothin is a bacterial metabolite that has been found in Streptomyces. It is an androgen receptor (AR) antagonist that inhibits binding of dihydrotestosterone (DHT) to ARs (IC50 = 13 μM) and inhibits DHT-induced exp... | |||
T68045 | Cioteronel | ||
Cioteronel is an antineoplastic compound with antiandrogenic activities. The antineoplastic action of CPC 10997 appears to be the inhibition of RNA synthesis in vitro. Although it blocks competitively the binding of dihy... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4000 | (±)-Equol | Equol,(R,S)-Equol | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Drug Metabolite |
(±)-Equol ((R,S)-Equol) is a non-steroidal estrogen produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. The estrogen receptor (ER) agonist activity of the naturally occu... | |||
T6491 | (-)-(S)-Equol | (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite |
(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-00932 | Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli |
Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli. |